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03-26
2022Dacomitinib (PF299804, PF299), CAS:1110813-31-4 大包装
Name:Dacomitinib (PF299804, PF299)Formulation:in 10mM DMSOTarget:EGFRPathway:Protein Tyrosine KinaseInformation:Dacomitinib (PF299804, PF299) is a potent, -
03-26
2022Fedratinib (SAR302503, TG101348), CAS:936091-26-8 工艺放大
Name:Fedratinib (SAR302503, TG101348)Formulation:in 10mM DMSOTarget:JAKPathway:JAK/STATInformation:Fedratinib (SAR302503, TG101348) is a selective inhibito -
03-26
2022Niraparib (MK-4827), CAS:1038915-60-4 线路优化
Name:Niraparib (MK-4827)Formulation:in 10mM DMSOTarget:PARPPathway:DNA DamageInformation:Niraparib (MK-4827) is a selective inhibitor of PARP1/2 with IC50 -
03-26
2022Canagliflozin, CAS:842133-18-0 化合物优化
Name:CanagliflozinFormulation:in 10mM DMSOTarget:SGLTPathway:GPCR & G ProteinInformation:Canagliflozin is a highly potent and selective SGLT2 inhibitor for -
03-26
2022Alectinib (CH5424802), CAS:1256580-46-7 公斤级
Name:Alectinib (CH5424802)Formulation:in 10mM DMSOTarget:ALKPathway:Protein Tyrosine KinaseInformation:Alectinib (CH5424802) is a potent ALK inhibitor with -
03-26
2022Tofacitinib (CP-690550,Tasocitinib), CAS:477600-75-2 小试供应
Name:Tofacitinib (CP-690550,Tasocitinib)Formulation:in 10mM DMSOTarget:JAKPathway:JAK/STATInformation:Tofacitinib (CP-690550,Tasocitinib) is a novel inhibi -
03-26
2022Istradefylline, CAS:155270-99-8 中试供应
Name:IstradefyllineFormulation:in 10mM DMSOTarget:Adenosine ReceptorPathway:GPCR & G ProteinInformation:Istradefylline is a selective adenosine A2A recepto -
03-26
2022Torcetrapib, CAS:262352-17-0 路线研究
Name:TorcetrapibFormulation:in 10mM DMSOTarget:CETPPathway:MetabolismInformation:Torcetrapib is a CETP inhibitor with IC50 of 37 nM, elevates HDL-C and red -
03-26
2022Lonafarnib, CAS:193275-84-2 化合物合成
Name:LonafarnibFormulation:in 10mM DMSOTarget:TransferasePathway:MetabolismInformation:Lonafarnib is an orally bioavailable FPTase inhibitor for H-ras, K-r -
03-26
2022Dabrafenib (GSK2118436), CAS:1195765-45-7 工艺优化
Name:Dabrafenib (GSK2118436)Formulation:in 10mM DMSOTarget:RafPathway:MAPKInformation:Dabrafenib (GSK2118436) is a mutant BRAFV600 specific inhibitor with


