-
03-26
2022Istradefylline, CAS:155270-99-8 中试供应
Name:IstradefyllineFormulation:in 10mM DMSOTarget:Adenosine ReceptorPathway:GPCR & G ProteinInformation:Istradefylline is a selective adenosine A2A recepto -
03-26
2022Torcetrapib, CAS:262352-17-0 路线研究
Name:TorcetrapibFormulation:in 10mM DMSOTarget:CETPPathway:MetabolismInformation:Torcetrapib is a CETP inhibitor with IC50 of 37 nM, elevates HDL-C and red -
03-26
2022Lonafarnib, CAS:193275-84-2 化合物合成
Name:LonafarnibFormulation:in 10mM DMSOTarget:TransferasePathway:MetabolismInformation:Lonafarnib is an orally bioavailable FPTase inhibitor for H-ras, K-r -
03-26
2022Dabrafenib (GSK2118436), CAS:1195765-45-7 工艺优化
Name:Dabrafenib (GSK2118436)Formulation:in 10mM DMSOTarget:RafPathway:MAPKInformation:Dabrafenib (GSK2118436) is a mutant BRAFV600 specific inhibitor with -
03-26
2022MPEP, CAS:96206-92-7 批量合成
Name:MPEPFormulation:in 10mM DMSOTarget:GluRPathway:Neuronal SignalingInformation:MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibit -
03-26
2022Alpelisib (BYL719), CAS:1217486-61-7 原料药研发
Name:Alpelisib (BYL719)Formulation:in 10mM DMSOTarget:PI3KPathway:PI3K/Akt/mTORInformation:Alpelisib (BYL719) is a potent and selective PI3Kα inhibitor wit -
03-26
2022Apalutamide?(ARN-509), CAS:956104-40-8 药物分子开发
Name:Apalutamide?(ARN-509)Formulation:in 10mM DMSOTarget:Androgen ReceptorPathway:Endocrinology & HormonesInformation:Apalutamide (ARN-509) is a selective -
03-26
2022Baricitinib (LY3009104, INCB028050), CAS:1187594-09-7 原研药中间体供应
Name:Baricitinib (LY3009104, INCB028050)Formulation:in 10mM DMSOTarget:JAKPathway:JAK/STATInformation:Baricitinib (LY3009104, INCB028050) is a selective JA -
03-26
2022Carfilzomib (PR-171), CAS:868540-17-4 新药中间体工艺
Name:Carfilzomib (PR-171)Formulation:in 10mM DMSOTarget:ProteasomePathway:ProteasesInformation:Carfilzomib (PR-171) is an irreversible proteasome inhibitor -
03-26
2022Alogliptin(SYK-322)benzoate, CAS:850649-62-6 新药中间体KG级
Name:Alogliptin(SYK-322)benzoateFormulation:in 10mM DMSOTarget:DPP-4Pathway:ProteasesInformation:Alogliptin is a potent, selective inhibitor of DPP-4 with