-
03-26
2022Clinofibrate, CAS:30299-08-2 新药中间体放大
Name:ClinofibrateFormulation:in 10mM DMSOTarget:HMG-CoA ReductasePathway:MetabolismInformation:Clinofibrate inhibits hydroxymethylglutaryl coenzyme A reduc -
03-26
2022Ciprofibrate, CAS:52214-84-3 线路优化
Name:CiprofibrateFormulation:in 10mM DMSOTarget:PPARPathway:DNA DamageInformation:Ciprofibrate is a peroxisome proliferator-activated receptor agonist.M.w. -
03-26
2022Trametinib (GSK1120212), CAS:871700-17-3 化合物优化
Name:Trametinib (GSK1120212)Formulation:in 10mM DMSOTarget:MEKPathway:MAPKInformation:Trametinib (GSK1120212) is a highly specific and potent MEK1/2 inhibi -
03-26
2022Ibrutinib (PCI-32765), CAS:936563-96-1 公斤级中间体
Name:Ibrutinib (PCI-32765)Formulation:in 10mM DMSOTarget:BTKPathway:AngiogenesisInformation:Ibrutinib (PCI-32765) is a potent and highly selective Brutons -
03-26
2022Dacomitinib (PF299804, PF299), CAS:1110813-31-4 大包装
Name:Dacomitinib (PF299804, PF299)Formulation:in 10mM DMSOTarget:EGFRPathway:Protein Tyrosine KinaseInformation:Dacomitinib (PF299804, PF299) is a potent, -
03-26
2022Fedratinib (SAR302503, TG101348), CAS:936091-26-8 工艺放大
Name:Fedratinib (SAR302503, TG101348)Formulation:in 10mM DMSOTarget:JAKPathway:JAK/STATInformation:Fedratinib (SAR302503, TG101348) is a selective inhibito -
03-26
2022Niraparib (MK-4827), CAS:1038915-60-4 线路优化
Name:Niraparib (MK-4827)Formulation:in 10mM DMSOTarget:PARPPathway:DNA DamageInformation:Niraparib (MK-4827) is a selective inhibitor of PARP1/2 with IC50 -
03-26
2022Canagliflozin, CAS:842133-18-0 化合物优化
Name:CanagliflozinFormulation:in 10mM DMSOTarget:SGLTPathway:GPCR & G ProteinInformation:Canagliflozin is a highly potent and selective SGLT2 inhibitor for -
03-26
2022Alectinib (CH5424802), CAS:1256580-46-7 公斤级
Name:Alectinib (CH5424802)Formulation:in 10mM DMSOTarget:ALKPathway:Protein Tyrosine KinaseInformation:Alectinib (CH5424802) is a potent ALK inhibitor with -
03-26
2022Tofacitinib (CP-690550,Tasocitinib), CAS:477600-75-2 小试供应
Name:Tofacitinib (CP-690550,Tasocitinib)Formulation:in 10mM DMSOTarget:JAKPathway:JAK/STATInformation:Tofacitinib (CP-690550,Tasocitinib) is a novel inhibi